Peer-reviewed veterinary case report
Identification of aminopiperidine benzamides as MCHr1 antagonists.
- Journal:
- Bioorganic & medicinal chemistry letters
- Year:
- 2005
- Authors:
- Vasudevan, Anil et al.
- Affiliation:
- Metabolic Diseases Research · United States
- Species:
- rodent
Abstract
The identification of a novel series of benzamide-containing MCHr1 antagonists is described. Compound 22 displayed moderate efficacy in a diet induced obesity mice model.
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Search related cases →Original publication: https://pubmed.ncbi.nlm.nih.gov/15950463/